6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-2,3,9-triMethyl-, (6S)-
- CasNo:202592-23-2
Product Description
Quality products?make an important contribution to long-term revenue and profitability. Reputable supplier selling 6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-2,3,9-triMethyl-, (6S)- 202592-23-2 with stock
1.What is the 6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-2,3,9-triMethyl-, (6S)- ?
(+)-JQ1 Carboxylic Acid is a selective inhibitor of BET bromodomains.
-
-
916489-36-6
methyl 2-((6S,Z)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f] [1,2,4]triazolo[4,3-a] [1,4]diazepin-6-yl)acetate
-
-
202592-23-2
(S)-[4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl]acetic acid
| Conditions | Yield |
|---|---|
|
With
lithium hydroxide monohydrate;
In
methanol;
at 20 ℃;
for 3h;
|
87%
|
|
With
methanol; lithium hydroxide monohydrate;
at 20 ℃;
for 3h;
|
87%
|
|
With
lithium hydroxide monohydrate;
In
methanol;
at 20 ℃;
for 3h;
|
87%
|
|
With
lithium hydroxide monohydrate; water;
In
methanol;
at 20 ℃;
for 3h;
|
87%
|
|
With
lithium hydroxide monohydrate;
In
methanol;
at 20 ℃;
for 3h;
|
87%
|
|
methyl 2-((6S,Z)-4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f] [1,2,4]triazolo[4,3-a] [1,4]diazepin-6-yl)acetate;
With
lithium hydroxide monohydrate; water;
In
methanol;
at 20 ℃;
for 3h;
With
hydrogenchloride;
In
water;
|
87%
|
|
With
lithium hydroxide monohydrate;
In
methanol;
at 20 ℃;
for 3h;
|
87%
|
|
With
lithium hydroxide monohydrate;
In
methanol;
at 20 ℃;
for 3h;
|
87%
|
|
With
methanol; lithium hydroxide monohydrate;
at 20 ℃;
for 3h;
|
87%
|
|
With
lithium hydroxide monohydrate;
In
methanol;
at 20 ℃;
for 3h;
|
87%
|
|
With
lithium hydroxide monohydrate;
In
methanol; water;
at 20 ℃;
for 3h;
Inert atmosphere;
|
87%
|
|
With
methanol; lithium hydroxide;
at 20 ℃;
for 3h;
|
87%
|
|
With
lithium hydroxide monohydrate;
In
methanol;
at 20 ℃;
for 2h;
|
87%
|
|
With
lithium hydroxide monohydrate; water;
In
methanol;
at 20 ℃;
for 3h;
|
87%
|
|
With
methanol; lithium hydroxide monohydrate;
at 20 ℃;
for 3h;
|
87%
|
|
With
lithium hydroxide monohydrate;
In
methanol;
at 20 ℃;
for 3h;
|
87%
|
|
With
water; sodium hydroxide;
In
methanol;
at 40 ℃;
for 1h;
|
-
-
1268524-70-4
(S)-tert-butyl 2-(4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)acetate
-
-
202592-23-2
(S)-[4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl]acetic acid
| Conditions | Yield |
|---|---|
|
With
formic acid;
at 20 ℃;
for 75h;
|
100%
|
|
With
formic acid;
at 20 ℃;
for 75h;
|
100%
|
|
With
trifluoroacetic acid;
In
dichloromethane;
at 20 ℃;
for 5h;
|
100%
|
|
With
formic acid;
for 48h;
Inert atmosphere;
|
99%
|
|
With
formic acid;
|
99%
|
|
With
trifluoroacetic acid;
at 20 ℃;
for 0.5h;
|
97%
|
|
With
trifluoroacetic acid;
In
dichloromethane;
at 23 ℃;
for 1h;
|
97%
|
|
With
formic acid;
at 25 ℃;
for 18h;
|
96%
|
|
With
formic acid;
at 25 ℃;
for 18h;
|
96%
|
|
In
dichloromethane;
at 20 ℃;
Acidic conditions;
|
96%
|
|
With
formic acid;
at 25 ℃;
for 12h;
|
96%
|
|
With
trifluoroacetic acid;
In
dichloromethane;
at 20 ℃;
|
95%
|
|
With
water; sodium hydroxide;
In
ethanol;
at 100 ℃;
for 2h;
|
94%
|
|
With
trifluoroacetic acid;
In
dichloromethane;
at 20 ℃;
for 7h;
|
93%
|
|
With
trifluoroacetic acid;
In
dichloromethane;
at 20 ℃;
for 2h;
|
90.1%
|
|
With
trifluoroacetic acid;
at 20 ℃;
for 4h;
|
76%
|
|
With
formic acid;
at 23 ℃;
|
|
|
With
formic acid;
at 20 ℃;
for 75h;
|
|
|
With
formic acid;
|
|
|
With
formic acid;
at 23 ℃;
for 72h;
|
|
|
With
formic acid;
In
formic acid;
for 96h;
|
|
|
With
formic acid;
at 20 ℃;
for 75h;
|
|
|
(S)-tert-butyl 2-(4-(4-chlorophenyl)-2,3,9-trimethyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepin-6-yl)acetate;
With
trifluoroacetic acid;
at 20 ℃;
for 2h;
With
sulfuric acid; sodium hydroxide;
In
tert-butyl methyl ether; water;
for 0.3h;
pH=7.3 - 7.5;
|
10.4 g
|
|
With
formic acid;
at 23 ℃;
for 72h;
|
|
|
With
trifluoroacetic acid;
In
dichloromethane;
|
|
|
With
trifluoroacetic acid;
In
chloroform;
at 40 ℃;
for 16h;
|
78 mg
|
|
With
formic acid;
at 20 ℃;
for 72h;
|
|
|
With
trifluoroacetic acid;
In
dichloromethane;
at 20 ℃;
for 2h;
|
|
|
With
trifluoroacetic acid;
In
dichloromethane;
|
|
|
With
trifluoroacetic acid;
In
dichloromethane;
at 20 ℃;
for 4h;
|
|
|
With
trifluoroacetic acid;
In
dichloromethane;
at 0 - 20 ℃;
for 16h;
Inert atmosphere;
|
|
|
With
trifluoroacetic acid;
In
dichloromethane;
at 20 ℃;
for 4h;
|
|
|
With
formic acid; trifluoroacetic acid;
In
dichloromethane;
at 15 ℃;
for 36h;
|
|
|
With
formic acid; trifluoroacetic acid;
In
dichloromethane;
at 15 ℃;
for 36h;
|
2.What is the CAS number for 6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-2,3,9-triMethyl-, (6S)- ?
The CAS number of 6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-2,3,9-triMethyl-, (6S)- is 202592-23-2.
More information of 6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-2,3,9-triMethyl-, (6S)- 202592-23-2 are:
|
CAS?Number |
202592-23-2 |
|
Density |
1.51±0.1 g/cm3(Predicted) |
|
Boiling Point |
661.6±65.0 °C(Predicted) |
|
PSA |
108.61000 |
|
LogP |
3.70980 |
|
Pka |
4.11±0.10(Predicted) |
3.What are another words for 6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-2,3,9-triMethyl-, (6S)- ?
Synonyms?for?6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-2,3,9-triMethyl-, (6S)- 202592-23-2:6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-2,3,9-triMethyl-, (6S)-;JQ-1 (carboxylic acid)
4.What is the molecular formula of 6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-2,3,9-triMethyl-, (6S)-?
The chemical formula of ?6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-2,3,9-triMethyl-, (6S)- is?C19 H17 ClN4 O2 S which containing 19 Carbon atoms,17 Hydrogen atoms,1 Chlorine atoms,4 Nitrogen atoms,2 Oxygen atoms and 1 Sulfur atoms,and the molecular weight of??6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-2,3,9-triMethyl-, (6S)-?is 400.889.
5.What is 6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-2,3,9-triMethyl-, (6S)- (202592-23-2) used for?
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6.Buy 6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-2,3,9-triMethyl-, (6S)- with the best price .
Shanghai Huachu Industrial Co. Ltd is a quality supplier of 6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-2,3,9-triMethyl-, (6S)-. Our main goal is customer satisfaction. Contact us to negotiate the best price for your business on 6H-Thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine-6-acetic acid, 4-(4-chlorophenyl)-2,3,9-triMethyl-, (6S)- 202592-23-2.